BDBM50442657 CHEMBL2442017

SMILES CCN([C@@H]1CCC[C@H](N)C1)C(=O)c1ccccc1OCc1ccccc1Cl

InChI Key InChIKey=MEZSPRSWKZUORF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442657   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50442657(CHEMBL2442017)Copy SMILESCopy InChI

Affinity DataIC50: 30nMAssay Description:Inhibition of human TRPM8 (unknown origin) expressed in HEK293 cells assessed as inhibition of WS12-induced Ca2+ elevation by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
4/13/2014
Entry Details Article
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