BDBM50442651 CHEMBL2442011

SMILES CCN(C1CCCC(N)C1)C(=O)c1ccccc1OCc1cccc(c1)C#N

InChI Key InChIKey=UNOZLBRAPWGPEZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442651   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50442651(CHEMBL2442011)Copy SMILESCopy InChI

Affinity DataIC50: 493nMAssay Description:Inhibition of human TRPM8 (unknown origin) expressed in HEK293 cells assessed as inhibition of WS12-induced Ca2+ elevation by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
4/13/2014
Entry Details Article
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