BDBM50442171 CHEMBL2441337

SMILES Cn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccnc2)c2c(N)ncnc12

InChI Key InChIKey=LIALAVDKTOKTGT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442171   

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50442171(CHEMBL2441337)Copy SMILESCopy InChI

Affinity DataIC50: 23nMAssay Description:Inhibition of GST-tagged PERK cytoplasmic domain (536 to 1116) (unknown origin) assessed as biotinylated His6-tagged EIF2alpha phosphorylation preinc...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
4/13/2014
Entry Details Article
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