BDBM50439415 CHEMBL2420549

SMILES CN(C)S(=O)(=O)c1cc(NC(=O)Nc2cccc(c2)C#N)ccc1C

InChI Key InChIKey=PLJCMVQIRQRQES-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50439415   

TargetG protein-activated inward rectifier potassium channel 4(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439415(CHEMBL2420549)
Affinity DataEC50:  3.30E+3nMAssay Description:Activation of GIRK1/4 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 1(Human)
Vanderbilt University

Curated by ChEMBL
LigandPNGBDBM50439415(CHEMBL2420549)
Affinity DataEC50:  3.90E+3nMAssay Description:Activation of GIRK1/2 (unknown origin) transfected in HEK293 cells after 4 mins by thallium flux-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed