BDBM50382252 CHEMBL2024502

SMILES CS(=O)(=O)Nc1ccc2cccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)c2c1

InChI Key InChIKey=WKJIKPBZHFHDBH-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50382252   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Bayer Yakuhin

Curated by ChEMBL

LigandBDBM50382252(CHEMBL2024502)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
Entry Details Article
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