BDBM50382244 CHEMBL2024493

SMILES Oc1cccc2c(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cccc12

InChI Key InChIKey=VEFWZCRRVABLLY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50382244   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Bayer Yakuhin

Curated by ChEMBL

LigandBDBM50382244(CHEMBL2024493)Copy SMILESCopy InChI

Affinity DataIC50: 45nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
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