BDBM50362095 CHEMBL1738942
SMILES CC(C)(C)c1cc(NC(=O)Nc2nccs2)n(n1)-c1ccc(CC(O)=O)cc1
InChI Key InChIKey=RBPOVRMRESQJOZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50362095
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataIC50: 9.17E+3nMAssay Description:Inhibition of wild type DDR2 (unknown origin) preincubated for 30 mins before substrate addition by FRET assayMore data for this Ligand-Target Pair
TargetDiscoidin domain-containing receptor 2(Human)
Technical University of Dortmund
Curated by ChEMBL
Technical University of Dortmund
Curated by ChEMBL
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity to human acrylodan-labeled N-terminal His-tagged DDR2 (558 to 855 aa) by FLiK assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Human)
Chemical Genomics Centre of The Max Planck Society
Curated by ChEMBL
Chemical Genomics Centre of The Max Planck Society
Curated by ChEMBL
Affinity DataKd: 196nMAssay Description:Binding affinity to N-terminus His-tagged human p38alpha expressed in Escherichia coli BL21 DE3 after 5 hrs by fluorescence analysisMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Human)
Chemical Genomics Centre of The Max Planck Society
Curated by ChEMBL
Chemical Genomics Centre of The Max Planck Society
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of N-terminus His-tagged human p38alpha expressed in Escherichia coli BL21 DE3 using GST-tagged ATF2 as substrate after 90 mins by HTRF as...More data for this Ligand-Target Pair