BDBM50359373 CHEMBL1929394

SMILES Cc1nc2cc(nn2c(C)c1C(=O)NCC(C)(C)NCC(=O)N1CCC[C@H]1C#N)-c1ccccc1

InChI Key InChIKey=FEFCYILNMDAYPD-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50359373   

TargetDipeptidyl peptidase 4(Human)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50359373(CHEMBL1929394)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant DPP-4 using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition measured after 20 mins by f...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50359373(CHEMBL1929394)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant DPP-8 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sanwa Kagaku Kenkyusho

Curated by ChEMBL
LigandPNGBDBM50359373(CHEMBL1929394)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed