BindingDB BDBM50359359 CHEMBL1929238

BDBM50359359 CHEMBL1929238

SMILES CN(C)CCN1CCN(CCC1=O)C(=O)c1cc(sc1NC(=O)Nc1cccc(Cl)c1Cl)C(C)(C)C

InChI Key InChIKey=SIUIQMQVKUUQQF-UHFFFAOYSA-N

Data 148 IC50

PDB links: 1 PDB ID matches this monomer.

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 148 hits for monomerid = 50359359

Cyclin-T1/Cyclin-dependent kinase 9(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK9/cyclin T1More data for this Ligand-Target Pair

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Protein kinase C beta type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.20E+4nMAssay Description:Inhibition of PKCbeta2More data for this Ligand-Target Pair

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Serine/threonine-protein kinase Chk1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair

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Cyclin-dependent kinase 5 activator 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK5/p35More data for this Ligand-Target Pair

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Misshapen-like kinase 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of MINKMore data for this Ligand-Target Pair

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Protein kinase C alpha type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair

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Protein kinase C eta type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCetaMore data for this Ligand-Target Pair

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Rho-associated protein kinase 2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of ROCK-2More data for this Ligand-Target Pair

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Macrophage-stimulating protein receptor(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of RONMore data for this Ligand-Target Pair

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Insulin receptor(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of IRMore data for this Ligand-Target Pair

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Vascular endothelial growth factor receptor 3(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of FLT4More data for this Ligand-Target Pair

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Serine/threonine-protein kinase BRSK1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of BRSK1More data for this Ligand-Target Pair

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cGMP-dependent protein kinase 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKG1alphaMore data for this Ligand-Target Pair

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Calcium/calmodulin-dependent protein kinase type II subunit beta(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 2.70E+3nMAssay Description:Inhibition of CAMK2betaMore data for this Ligand-Target Pair

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cGMP-dependent protein kinase 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKG1betaMore data for this Ligand-Target Pair

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Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase 17A(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of DRAK1More data for this Ligand-Target Pair

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Mitogen-activated protein kinase 14(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 22nMAssay Description:Inhibition of p38alpha assessed as [33P]gamma-ATP incorporation into GST-ATF2 substrate preincubated for 20 mins before substrate addition measured a...More data for this Ligand-Target Pair

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3D Structure (crystal)

Cyclin-dependent kinase 5 activator 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair

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Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair

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Cyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CDK2/cyclin EMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase PAK 5(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PAK5More data for this Ligand-Target Pair

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Serine/threonine-protein kinase PAK 6(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PAK6More data for this Ligand-Target Pair

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PAS domain-containing serine/threonine-protein kinase(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PASKMore data for this Ligand-Target Pair

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Platelet-derived growth factor receptor alpha(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PDGFRalphaMore data for this Ligand-Target Pair

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Platelet-derived growth factor receptor beta(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair

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[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair

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Phosphorylase b kinase gamma catalytic chain, liver/testis isoform(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PHKgamma2More data for this Ligand-Target Pair

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Serine/threonine-protein kinase pim-1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair

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Serine/threonine-protein kinase pim-2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PIM2More data for this Ligand-Target Pair

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Protein kinase C beta type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCbeta1More data for this Ligand-Target Pair

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Protein kinase C delta type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 1.50E+4nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair

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Protein kinase C gamma type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCgammaMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase D1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCmuMore data for this Ligand-Target Pair

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Protein kinase C theta type(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair

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Polycystin-2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PKD2More data for this Ligand-Target Pair

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Serine/threonine-protein kinase PLK1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PLK1More data for this Ligand-Target Pair

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Serine/threonine-protein kinase PLK2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of PLK2More data for this Ligand-Target Pair

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Cytochrome P450 3A4(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 550nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair

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Tyrosine-protein kinase BTK(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of BTKMore data for this Ligand-Target Pair

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Calcium/calmodulin-dependent protein kinase type II subunit delta(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 1.20E+4nMAssay Description:Inhibition of CAMK2deltaMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase Chk2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CHK2More data for this Ligand-Target Pair

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Casein kinase I isoform alpha(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CK1More data for this Ligand-Target Pair

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Casein kinase II subunit alpha(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CK2alphaMore data for this Ligand-Target Pair

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Hepatocyte growth factor receptor(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of c-METMore data for this Ligand-Target Pair

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Tyrosine-protein kinase CSK(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of CSKMore data for this Ligand-Target Pair

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Proto-oncogene tyrosine-protein kinase Src(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair

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Death-associated protein kinase 1(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of DAPK1More data for this Ligand-Target Pair

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Discoidin domain-containing receptor 2(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 7.00E+3nMAssay Description:Inhibition of DDR2More data for this Ligand-Target Pair

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Epidermal growth factor receptor(Human)
Ansaris

Curated by ChEMBL

BDBM50359359(CHEMBL1929238)

IC50: 3.00E+4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair

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Displayed 1 to 50 (of 148 total ) | Next | Last >>

Filter my 148 hits

Targets 144▿
- Protein kinase C beta type 2
- cGMP-dependent protein kinase 1 2
- Mitogen-activated protein kinase 14 2
- Cyclin-dependent kinase 5 activator 1 2
- Mitogen-activated protein kinase 11/12/13/14 1
- Receptor tyrosine-protein kinase erbB-4 1
- Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 1
- Hepatocyte growth factor receptor 1
- ALK tyrosine kinase receptor 1
- Glycogen synthase kinase-3 beta 1
- NUAK family SNF1-like kinase 1 1
- Receptor-type tyrosine-protein kinase FLT3 1
- Calcium/calmodulin-dependent protein kinase type II subunit beta 1
- Serine/threonine-protein kinase Nek3 1
- Macrophage-stimulating protein receptor 1
- Protein kinase C theta type 1
- Homeodomain-interacting protein kinase 3 1
- Serine/threonine-protein kinase PAK 2 1
- Serine/threonine-protein kinase PAK 3 1
- Serine/threonine-protein kinase PAK 4 1
- Serine/threonine-protein kinase PAK 5 1
- Serine/threonine-protein kinase PAK 6 1
- Tyrosine-protein kinase JAK3 1
- Tyrosine-protein kinase JAK2 1
- Proto-oncogene tyrosine-protein kinase receptor Ret 1
- Tyrosine-protein kinase ZAP-70 1
- Serine/threonine-protein kinase Sgk1 1
- Ephrin type-A receptor 1 1
- Ephrin type-A receptor 3 1
- Ephrin type-A receptor 2 1
- Ephrin type-A receptor 5 1
- Tyrosine-protein kinase BTK 1
- Ephrin type-A receptor 4 1
- Tyrosine-protein kinase receptor UFO 1
- Protein kinase C eta type 1
- Insulin-like growth factor 1 receptor 1
- Tyrosine-protein kinase Blk 1
- Receptor-interacting serine/threonine-protein kinase 2 1
- Epidermal growth factor receptor 1
- Serine/threonine-protein kinase NLK 1
- Homeodomain-interacting protein kinase 1 1
- Ribosomal protein S6 kinase beta-1 1
- Tyrosine-protein kinase Lyn 1
- Focal adhesion kinase 1 1
- Ephrin type-B receptor 3 1
- Serine/threonine-protein kinase 33 1
- Ephrin type-B receptor 4 1
- Ephrin type-B receptor 1 1
- Ephrin type-B receptor 2 1
- MAP kinase-activated protein kinase 2 1
- MAP kinase-activated protein kinase 3 1
- Platelet-derived growth factor receptor beta 1
- MAP kinase-activated protein kinase 5 1
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial 1
- Death-associated protein kinase 1 1
- Tyrosine-protein kinase Fer 1
- Serine/threonine-protein kinase D1 1
- Calcium/calmodulin-dependent protein kinase type II subunit delta 1
- PAS domain-containing serine/threonine-protein kinase 1
- Death-associated protein kinase 3 1
- Proto-oncogene tyrosine-protein kinase ROS 1
- Serine/threonine-protein kinase pim-1 1
- Serine/threonine-protein kinase pim-2 1
- Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2 1
- Angiopoietin-1 receptor 1
- Testis-specific serine/threonine-protein kinase 2 1
- Protein-tyrosine kinase 6 1
- Activin receptor type-1B 1
- Casein kinase II subunit alpha 1
- Interleukin-1 receptor-associated kinase 4 1
- Cytoplasmic tyrosine-protein kinase BMX 1
- Mitogen-activated protein kinase kinase kinase 9 1
- RAC-gamma serine/threonine-protein kinase 1
- Mitogen-activated protein kinase kinase kinase 5 1
- Interleukin-1 receptor-associated kinase 1 1
- Tyrosine-protein kinase ABL2 1
- Tyrosine-protein kinase ABL1 1
- RAC-alpha serine/threonine-protein kinase 1
- Rho-associated protein kinase 2 1
- Rho-associated protein kinase 1 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Tyrosine-protein kinase Fes/Fps 1
- BDNF/NT-3 growth factors receptor 1
- Mitogen-activated protein kinase 1 1
- Serine/threonine-protein kinase 3 1
- Serine/threonine-protein kinase 17A 1
- Tyrosine-protein kinase Lck 1
- Mitogen-activated protein kinase 3 1
- Discoidin domain-containing receptor 2 1
- Serine/threonine-protein kinase 4 1
- Protein kinase C delta type 1
- Mitogen-activated protein kinase 9 1
- G protein-coupled receptor kinase 5 1
- Protein-tyrosine kinase 2-beta 1
- High affinity nerve growth factor receptor 1
- G protein-coupled receptor kinase 6 1
- Mitogen-activated protein kinase 8 1
- Tyrosine-protein kinase SYK 1
- Ribosomal protein S6 kinase alpha-1 1
- Serine/threonine-protein kinase TBK1 1
- Cyclin-T1/Cyclin-dependent kinase 9 1
- Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 1
- Fibroblast growth factor receptor 4 1
- Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1 1
- Vascular endothelial growth factor receptor 2 1
- Tyrosine-protein kinase Fgr 1
- Insulin receptor 1
- Vascular endothelial growth factor receptor 3 1
- Tyrosine-protein kinase HCK 1
- Aurora kinase A 1
- Fibroblast growth factor receptor 1 1
- Fibroblast growth factor receptor 2 1
- Fibroblast growth factor receptor 3 1
- Vascular endothelial growth factor receptor 1 1
- Cytochrome P450 3A4 1
- Serine/threonine-protein kinase PLK1 1
- Insulin receptor-related protein 1
- Serine/threonine-protein kinase PLK2 1
- Inhibitor of nuclear factor kappa-B kinase subunit beta 1
- Serine/threonine-protein kinase PLK3 1
- Mitogen-activated protein kinase 13 1
- Mitogen-activated protein kinase 12 1
- Mitogen-activated protein kinase 11 1
- RAC-beta serine/threonine-protein kinase 1
- Mitogen-activated protein kinase 10 1
- Serine/threonine-protein kinase BRSK1 1
- Casein kinase I isoform alpha 1
- Protein kinase C gamma type 1
- Misshapen-like kinase 1 1
- Tyrosine-protein kinase Fyn 1
- Tyrosine-protein kinase CSK 1
- Macrophage colony-stimulating factor 1 receptor 1
- Protein kinase C alpha type 1
- Ribosomal protein S6 kinase alpha-4 1
- Platelet-derived growth factor receptor alpha 1
- Ribosomal protein S6 kinase alpha-5 1
- Serine/threonine-protein kinase Chk2 1
- Serine/threonine-protein kinase MARK1 1
- Serine/threonine-protein kinase MARK2 1
- Serine/threonine-protein kinase Chk1 1
- cAMP-dependent protein kinase catalytic subunit PRKX 1
- Polycystin-2 1
- Tyrosine-protein kinase Yes 1
- Serine/threonine-protein kinase WNK2 1
Publications 2▿
- Bioorg Med Chem Lett 21: 7155-65 (2011) 147
- Eur J Med Chem 143: 1616-1634 (2018) 1
Institutions 2▿
- Ansaris 147
- University of Zagreb 1
Affinity: 22 to 5.0E+4 nM▿
- IC50 148
- Affinity ≤ nM
Xtal structures: 1
Docked structures: 0
Catalog Cmpds: 0