BindingDB BDBM50326054 CHEMBL1240703

BDBM50326054 CHEMBL1240703

SMILES CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1

InChI Key InChIKey=ZZSBPGIGIUFJRA-UHFFFAOYSA-N

Data 1 IC50 359 Kd

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 360 hits for monomerid = 50326054

Mitogen-activated protein kinase kinase kinase 4(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MAP3K4More data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
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Tyrosine-protein kinase JAK1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to JAK1 JH2 domainMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Calcium/calmodulin-dependent protein kinase type II subunit beta(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to CAMK2BMore data for this Ligand-Target Pair

PDB KEGG
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Myosin light chain kinase, smooth muscle(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MLCKMore data for this Ligand-Target Pair

PDB KEGG
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SRSF protein kinase 3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 3.50E+3nMAssay Description:Binding affinity to SRPK3More data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
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Calcium/calmodulin-dependent protein kinase type II subunit gamma(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 2.60E+3nMAssay Description:Binding affinity to CAMK2GMore data for this Ligand-Target Pair

PDB KEGG
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Aurora kinase B(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 7.50E+5nMAssay Description:Binding affinity to AURKBMore data for this Ligand-Target Pair

PDB KEGG
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Ribosomal protein S6 kinase alpha-1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA4(Kin.Dom.1-N-terminal)More data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
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Serine/threonine-protein kinase 17A(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to DRAK1More data for this Ligand-Target Pair

PDB KEGG
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MAP/microtubule affinity-regulating kinase 3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 490nMAssay Description:Binding affinity to MARK3More data for this Ligand-Target Pair

PDB KEGG
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Ephrin type-A receptor 1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to EPHA1More data for this Ligand-Target Pair

UniProtKB/SwissProt
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Death-associated protein kinase 1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to DAPK1More data for this Ligand-Target Pair

PDB KEGG
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Vascular endothelial growth factor receptor 3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to FLT4More data for this Ligand-Target Pair

PDB KEGG
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SRSF protein kinase 2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to SRPK2More data for this Ligand-Target Pair

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Protein kinase C alpha type(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to PKAC-alphaMore data for this Ligand-Target Pair

PDB KEGG
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Protein kinase C eta type(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to PRKCHMore data for this Ligand-Target Pair

PDB KEGG
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Misshapen-like kinase 1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MINKMore data for this Ligand-Target Pair

PDB KEGG
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Interleukin-1 receptor-associated kinase 3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to IRAK3More data for this Ligand-Target Pair

PDB
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cGMP-dependent protein kinase 1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to PRKG1More data for this Ligand-Target Pair

PDB KEGG
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Rho-associated protein kinase 2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to ROCK2More data for this Ligand-Target Pair

PDB KEGG
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Serine/threonine-protein kinase D2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to PRKD2More data for this Ligand-Target Pair

PDB KEGG
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Serine/threonine-protein kinase MRCK gamma(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to DMPK2More data for this Ligand-Target Pair

KEGG
UniProtKB/SwissProt
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Ephrin type-A receptor 6(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to EPHA6More data for this Ligand-Target Pair

KEGG
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Ribosomal protein S6 kinase alpha-6(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA6(Kin.Dom.2-C-terminal)More data for this Ligand-Target Pair

PDB KEGG
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Serine/threonine-protein kinase DCLK2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to DCAMKL2More data for this Ligand-Target Pair

PDB KEGG
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Serine/threonine-protein kinase Chk1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 3.50E+5nMAssay Description:Binding affinity to CHEK1More data for this Ligand-Target Pair

PDB KEGG
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Cyclin-dependent kinase 11A(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to CDC2L2More data for this Ligand-Target Pair

PDB KEGG
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Myosin-IIIb(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MYO3BMore data for this Ligand-Target Pair

KEGG
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Serine/threonine-protein kinase BRSK1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to BRSK1More data for this Ligand-Target Pair

PDB KEGG
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Non-receptor tyrosine-protein kinase TYK2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to TYK2(JH2domain-pseudokinase)More data for this Ligand-Target Pair

PDB KEGG
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AP2-associated protein kinase 1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 960nMAssay Description:Binding affinity to AAK1More data for this Ligand-Target Pair

PDB KEGG
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Ribosomal protein S6 kinase alpha-4(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA1(Kin.Dom.2-C-terminal)More data for this Ligand-Target Pair

KEGG
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Inhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to IKK-alphaMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase TAO1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to TAOK1More data for this Ligand-Target Pair

PDB KEGG
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Cyclin-dependent kinase 15(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to PFTAIRE2More data for this Ligand-Target Pair

KEGG
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Receptor-type tyrosine-protein kinase FLT3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

IC50: 350nMAssay Description:Inhibition of FLT3 autophosphorylation in human RS4-11 cells after 2 hrs by electrochemiluminescence assayMore data for this Ligand-Target Pair

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Calcium/calmodulin-dependent protein kinase kinase 2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 790nMAssay Description:Binding affinity to CAMKK2More data for this Ligand-Target Pair

PDB KEGG
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Serine/threonine-protein kinase TNNI3K(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to TNNI3KMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase ULK2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to ULK2More data for this Ligand-Target Pair

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Ribosomal protein S6 kinase alpha-2(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA5(Kin.Dom.1-N-terminal)More data for this Ligand-Target Pair

PDB KEGG
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Calcium/calmodulin-dependent protein kinase type II subunit alpha(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 690nMAssay Description:Binding affinity to CAMK2AMore data for this Ligand-Target Pair

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Myosin light chain kinase, smooth muscle(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MYLKMore data for this Ligand-Target Pair

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Macrophage-stimulating protein receptor(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to MST1RMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase 35(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to STK35More data for this Ligand-Target Pair

KEGG
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Myotonin-protein kinase(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to DMPKMore data for this Ligand-Target Pair

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Mitogen-activated protein kinase kinase kinase 20(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to ZAKMore data for this Ligand-Target Pair

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Serine/threonine-protein kinase ULK1(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to ULK1More data for this Ligand-Target Pair

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Receptor-type tyrosine-protein kinase FLT3(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: 68nMAssay Description:Binding affinity to FLT3More data for this Ligand-Target Pair

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Hormonally up-regulated neu tumor-associated kinase(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to HUNKMore data for this Ligand-Target Pair

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Ribosomal protein S6 kinase alpha-5(Human)
Ambit Biosciences

Curated by ChEMBL

BDBM50326054(CHEMBL1240703)

Kd: >1.00E+4nMAssay Description:Binding affinity to RPS6KA2(Kin.Dom.2-C-terminal)More data for this Ligand-Target Pair

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Displayed 1 to 50 (of 360 total ) | Next | Last >>

Filter my 360 hits

Targets 346▿
- Receptor-type tyrosine-protein kinase FLT3 3
- Ribosomal protein S6 kinase alpha-2 2
- Ribosomal protein S6 kinase alpha-1 2
- Ephrin type-A receptor 6 2
- Non-receptor tyrosine-protein kinase TYK2 2
- Mitogen-activated protein kinase 14 2
- Myosin light chain kinase, smooth muscle 2
- Tyrosine-protein kinase JAK1 2
- Serine/threonine-protein kinase TAO1 2
- Ribosomal protein S6 kinase alpha-6 2
- Calcium/calmodulin-dependent protein kinase type II subunit gamma 2
- Ribosomal protein S6 kinase alpha-4 2
- Ribosomal protein S6 kinase alpha-5 2
- Tyrosine-protein kinase Tec 1
- BMP-2-inducible protein kinase 1
- Rhodopsin kinase GRK1 1
- Cyclin-dependent kinase 11B 1
- Cyclin-dependent kinase 11A 1
- Uncharacterized serine/threonine-protein kinase SBK3 1
- LIM domain kinase 1 1
- LIM domain kinase 2 1
- ALK tyrosine kinase receptor 1
- NUAK family SNF1-like kinase 2 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform 1
- Glycogen synthase kinase-3 beta 1
- Calcium/calmodulin-dependent protein kinase type 1 1
- NUAK family SNF1-like kinase 1 1
- AP2-associated protein kinase 1 1
- Calcium/calmodulin-dependent protein kinase type II subunit beta 1
- Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform 1
- Serine/threonine-protein kinase PAK 1 1
- Protein kinase C theta type 1
- Serine/threonine-protein kinase PAK 2 1
- Serine/threonine-protein kinase PAK 3 1
- Dual specificity mitogen-activated protein kinase kinase 2 1
- Serine/threonine-protein kinase PAK 4 1
- Phosphatidylinositol 5-phosphate 4-kinase type-2 beta 1
- Serine/threonine-protein kinase tousled-like 2 1
- Dual specificity mitogen-activated protein kinase kinase 3 1
- Serine/threonine-protein kinase PAK 5 1
- Serine/threonine-protein kinase PAK 6 1
- Serine/threonine-protein kinase tousled-like 1 1
- Tyrosine-protein kinase JAK3 1
- Tyrosine-protein kinase JAK2 1
- Dual specificity mitogen-activated protein kinase kinase 1 1
- Protein delta homolog 1 1
- Dual specificity mitogen-activated protein kinase kinase 6 1
- Dual specificity mitogen-activated protein kinase kinase 4 1
- Tyrosine-protein kinase ZAP-70 1
- Casein kinase I isoform gamma-3 1
- Casein kinase I isoform gamma-2 1
- Casein kinase I isoform epsilon 1
- Casein kinase I isoform gamma-1 1
- Ephrin type-A receptor 1 1
- Ephrin type-A receptor 3 1
- Ephrin type-A receptor 2 1
- Ephrin type-A receptor 5 1
- Tyrosine-protein kinase BTK 1
- Ephrin type-A receptor 4 1
- Tyrosine-protein kinase receptor UFO 1
- Insulin-like growth factor 1 receptor 1
- Activin receptor type-1 1
- Myosin light chain kinase 2, skeletal/cardiac muscle 1
- Tyrosine-protein kinase Srms 1
- Wee1-like protein kinase 1
- U4/U6 small nuclear ribonucleoprotein Prp4 1
- Serine/threonine-protein kinase/endoribonuclease IRE1 1
- Serine/threonine-protein kinase MAK 1
- Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma 1
- Ankyrin repeat and protein kinase domain-containing protein 1 1
- Tyrosine-protein kinase Lyn 1
- Focal adhesion kinase 1 1
- Cyclin-dependent kinase 2 1
- Tyrosine-protein kinase TXK 1
- Rhodopsin kinase GRK7 1
- Ephrin type-A receptor 8 1
- Phosphatidylinositol 4-kinase beta 1
- Death-associated protein kinase 2 1
- Death-associated protein kinase 1 1
- Serine/threonine-protein kinase D2 1
- Serine/threonine-protein kinase D3 1
- TGF-beta receptor type-2 1
- Serine/threonine-protein kinase D1 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 1
- Death-associated protein kinase 3 1
- Cyclin-dependent kinase 9 1
- Serine/threonine-protein kinase pim-3 1
- Cyclin-dependent kinase 8 1
- Cyclin-dependent kinase 7 1
- Serine/threonine-protein kinase pim-1 1
- Cyclin-dependent kinase 5 1
- Serine/threonine-protein kinase pim-2 1
- Serine/threonine-protein kinase 38 1
- Serine/threonine-protein kinase 35 1
- Cyclin-dependent kinase 3 1
- Serine/threonine-protein kinase 36 1
- Cyclin-dependent kinase 16 1
- Testis-specific serine/threonine-protein kinase 1 1
- Protein kinase C epsilon type 1
- Cyclin-dependent kinase 17 1
- Bone morphogenetic protein receptor type-2 1
- Cyclin-dependent kinase 19 1
- Protein-tyrosine kinase 6 1
- Casein kinase II subunit alpha 1
- Cyclin-dependent kinase 14 1
- Cyclin-dependent kinase 15 1
- Leukocyte tyrosine kinase receptor 1
- Cytoplasmic tyrosine-protein kinase BMX 1
- Tyrosine-protein kinase ABL2 1
- Tyrosine-protein kinase ABL1 1
- Atypical kinase COQ8B, mitochondrial 1
- Microtubule-associated serine/threonine-protein kinase 1 1
- Calcium/calmodulin-dependent protein kinase type II subunit alpha 1
- cGMP-dependent protein kinase 2 1
- Rho-associated protein kinase 2 1
- cGMP-dependent protein kinase 1 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 1
- Rho-associated protein kinase 1 1
- Serine/threonine-protein kinase ULK1 1
- Serine/threonine-protein kinase SIK2 1
- Tyrosine-protein kinase Fes/Fps 1
- Serine/threonine-protein kinase SIK1 1
- Serine/threonine-protein kinase ULK2 1
- Serine/threonine-protein kinase ULK3 1
- 3-phosphoinositide-dependent protein kinase 1 1
- Mitogen-activated protein kinase 1 1
- Serine/threonine-protein kinase 3 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform 1
- Mitogen-activated protein kinase 3 1
- Discoidin domain-containing receptor 2 1
- Mitogen-activated protein kinase 4 1
- Serine/threonine-protein kinase 4 1
- SRSF protein kinase 3 1
- Mitogen-activated protein kinase 9 1
- SRSF protein kinase 2 1
- Mitogen-activated protein kinase 6 1
- Mitogen-activated protein kinase 7 1
- Calcium/calmodulin-dependent protein kinase type IV 1
- Mitogen-activated protein kinase 8 1
- Tyrosine-protein kinase SYK 1
- Serine/threonine-protein kinase TBK1 1
- Serine/threonine-protein kinase RIO1 1
- Serine/threonine-protein kinase LATS1 1
- Serine/threonine-protein kinase RIO3 1
- Serine/threonine-protein kinase 32B 1
- Serine/threonine-protein kinase RIO2 1
- Serine/threonine-protein kinase 32C 1
- Vascular endothelial growth factor receptor 2 1
- Insulin receptor 1
- Tyrosine-protein kinase HCK 1
- Vascular endothelial growth factor receptor 3 1
- Vascular endothelial growth factor receptor 1 1
- Serine/threonine-protein kinase PLK1 1
- Serine/threonine-protein kinase PLK2 1
- Insulin receptor-related protein 1
- Inhibitor of nuclear factor kappa-B kinase subunit beta 1
- Serine/threonine-protein kinase NIM1 1
- Serine/threonine-protein kinase PLK3 1
- Serine/threonine-protein kinase PLK4 1
- Tyrosine-protein kinase receptor TYRO3 1
- Wee1-like protein kinase 2 1
- Serine/threonine-protein kinase BRSK1 1
- Serine/threonine-protein kinase LATS2 1
- Citron Rho-interacting kinase 1
- Platelet-derived growth factor receptor alpha 1
- Serine/threonine-protein kinase BRSK2 1
- Serine/threonine-protein kinase Chk2 1
- Serine/threonine-protein kinase Chk1 1
- cAMP-dependent protein kinase catalytic subunit PRKX 1
- SRSF protein kinase 1 1
- Tyrosine-protein kinase Yes 1
- Serine/threonine-protein kinase MRCK beta 1
- Serine/threonine-protein kinase MRCK gamma 1
- Casein kinase II subunit alpha' 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 2 1
- Serine/threonine-protein kinase STK11 1
- Cyclin-G-associated kinase 1
- Receptor tyrosine-protein kinase erbB-4 1
- Receptor tyrosine-protein kinase erbB-2 1
- Tyrosine-protein kinase FRK 1
- Receptor tyrosine-protein kinase erbB-3 1
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform 1
- Hepatocyte growth factor receptor 1
- Serine/threonine-protein kinase B-raf 1
- Serine/threonine-protein kinase Nek9 1
- Serine/threonine-protein kinase Nek7 1
- Glycogen synthase kinase-3 alpha 1
- Serine/threonine-protein kinase Nek6 1
- Serine/threonine-protein kinase Nek5 1
- Serine/threonine-protein kinase Nek2 1
- Serine/threonine-protein kinase receptor R3 1
- Serine/threonine-protein kinase Nek1 1
- Macrophage-stimulating protein receptor 1
- Cyclin-dependent kinase-like 3 1
- Serine/threonine-protein kinase SIK3 [59-1321] 1
- Cyclin-dependent kinase-like 2 1
- MAP/microtubule affinity-regulating kinase 3 1
- Homeodomain-interacting protein kinase 4 1
- Homeodomain-interacting protein kinase 3 1
- MAP kinase-interacting serine/threonine-protein kinase 2 1
- MAP kinase-interacting serine/threonine-protein kinase 1 1
- Cyclin-dependent kinase-like 5 1
- Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase 1
- Serine/threonine-protein kinase 10 1
- MAP/microtubule affinity-regulating kinase 4 1
- Proto-oncogene tyrosine-protein kinase receptor Ret 1
- Serine/threonine-protein kinase 38-like 1
- Dual specificity protein kinase TTK 1
- Myosin-IIIb 1
- Myosin-IIIa 1
- Tyrosine-protein kinase ITK/TSK 1
- Myotonin-protein kinase 1
- Protein kinase C eta type 1
- Bone morphogenetic protein receptor type-1B 1
- Bone morphogenetic protein receptor type-1A 1
- Tyrosine-protein kinase Blk 1
- Receptor-interacting serine/threonine-protein kinase 1 1
- Serine/threonine-protein kinase 16 1
- Receptor-interacting serine/threonine-protein kinase 2 1
- Epidermal growth factor receptor 1
- Non-receptor tyrosine-protein kinase TNK1 1
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon 1
- Serine/threonine-protein kinase NLK 1
- Homeodomain-interacting protein kinase 2 1
- Homeodomain-interacting protein kinase 1 1
- Receptor-interacting serine/threonine-protein kinase 4 1
- Ribosomal protein S6 kinase beta-1 1
- Serine/threonine-protein kinase OSR1 1
- Casein kinase I isoform delta 1
- Cyclin-dependent kinase 18 [3-474] 1
- RAF proto-oncogene serine/threonine-protein kinase 1
- Serine/threonine-protein kinase 26 1
- Serine/threonine-protein kinase 24 1
- Serine/threonine-protein kinase 25 1
- Dual specificity testis-specific protein kinase 1 1
- Ephrin type-B receptor 3 1
- Serine/threonine-protein kinase 33 1
- Ephrin type-B receptor 4 1
- Ephrin type-B receptor 1 1
- Ephrin type-B receptor 2 1
- MAP kinase-activated protein kinase 2 1
- Ephrin type-B receptor 6 1
- Platelet-derived growth factor receptor beta 1
- Epithelial discoidin domain-containing receptor 1 1
- MAP kinase-activated protein kinase 5 1
- STE20/SPS1-related proline-alanine-rich protein kinase 1
- Muscle, skeletal receptor tyrosine-protein kinase 1
- Tyrosine-protein kinase Fer 1
- Tyrosine-protein kinase receptor Tie-1 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-2 1
- Calcium/calmodulin-dependent protein kinase type II subunit delta 1
- Proto-oncogene tyrosine-protein kinase ROS 1
- Serine/threonine-protein kinase DCLK1 1
- Calcium/calmodulin-dependent protein kinase kinase 1 1
- Serine/threonine-protein kinase DCLK2 1
- Serine/threonine-protein kinase TAO3 1
- Calcium/calmodulin-dependent protein kinase kinase 2 1
- Serine/threonine-protein kinase DCLK3 1
- Serine/threonine-protein kinase TNNI3K 1
- Interferon-induced, double-stranded RNA-activated protein kinase 1
- Angiopoietin-1 receptor 1
- Mitogen-activated protein kinase kinase kinase kinase 2 1
- Mitogen-activated protein kinase kinase kinase kinase 3 1
- Mast/stem cell growth factor receptor Kit 1
- Mitogen-activated protein kinase kinase kinase kinase 1 1
- Serine/threonine-protein kinase MRCK alpha 1
- Mitogen-activated protein kinase kinase kinase kinase 4 1
- Mitogen-activated protein kinase kinase kinase kinase 5 1
- Mitogen-activated protein kinase 15 1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1 1
- Activin receptor type-1B 1
- Myosin light chain kinase family member 4 1
- Mitogen-activated protein kinase kinase kinase 9 1
- Mitogen-activated protein kinase kinase kinase 6 1
- RAC-gamma serine/threonine-protein kinase 1
- Mitogen-activated protein kinase kinase kinase 5 1
- Interleukin-1 receptor-associated kinase 1 1
- Mitogen-activated protein kinase kinase kinase 7 1
- Interleukin-1 receptor-associated kinase 3 1
- Mitogen-activated protein kinase kinase kinase 2 1
- Mitogen-activated protein kinase kinase kinase 1 1
- Mitogen-activated protein kinase kinase kinase 4 1
- Mitogen-activated protein kinase kinase kinase 3 1
- Serine/threonine-protein kinase ICK 1
- RAC-alpha serine/threonine-protein kinase 1
- Megakaryocyte-associated tyrosine-protein kinase 1
- Proto-oncogene tyrosine-protein kinase Src 1
- Activin receptor type-2B 1
- Activin receptor type-2A 1
- BDNF/NT-3 growth factors receptor 1
- Serine/threonine-protein kinase 17A 1
- Tyrosine-protein kinase Lck 1
- Serine/threonine-protein kinase 17B 1
- Mitogen-activated protein kinase kinase kinase 19 1
- Dual specificity protein kinase CLK1 1
- Protein kinase C delta type 1
- Mitogen-activated protein kinase kinase kinase 15 1
- NT-3 growth factor receptor 1
- G protein-coupled receptor kinase 4 1
- Dual specificity protein kinase CLK4 1
- Dual specificity protein kinase CLK3 1
- Dual specificity protein kinase CLK2 1
- High affinity nerve growth factor receptor 1
- Protein-tyrosine kinase 2-beta 1
- Tyrosine-protein kinase Mer 1
- Poly [ADP-ribose] polymerase tankyrase-2 1
- Serine/threonine-protein kinase N2 1
- cAMP-dependent protein kinase catalytic subunit beta 1
- Serine/threonine-protein kinase N1 1
- Ribosomal protein S6 kinase alpha-3 1
- Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 1
- Calcium/calmodulin-dependent protein kinase type 1D 1
- STE20-like serine/threonine-protein kinase 1
- Hormonally up-regulated neu tumor-associated kinase 1
- Fibroblast growth factor receptor 4 1
- Tyrosine-protein kinase Fgr 1
- Aurora kinase B 1
- Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta 1
- Aurora kinase A 1
- Mitogen-activated protein kinase kinase kinase 20 1
- Fibroblast growth factor receptor 1 1
- Fibroblast growth factor receptor 2 1
- Atypical kinase COQ8A, mitochondrial 1
- Fibroblast growth factor receptor 3 1
- Aurora kinase C 1
- Mitogen-activated protein kinase 13 1
- Inhibitor of nuclear factor kappa-B kinase subunit alpha 1
- Mitogen-activated protein kinase 12 1
- Mitogen-activated protein kinase 11 1
- Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha 1
- RAC-beta serine/threonine-protein kinase 1
- Mitogen-activated protein kinase 10 1
- Casein kinase I isoform alpha 1
- Misshapen-like kinase 1 1
- Tyrosine-protein kinase Fyn 1
- Tyrosine-protein kinase CSK 1
- Macrophage colony-stimulating factor 1 receptor 1
- Protein kinase C alpha type 1
- Maternal embryonic leucine zipper kinase 1
- Serine/threonine-protein kinase MARK1 1
- Serine/threonine-protein kinase MARK2 1
- TRAF2 and NCK-interacting protein kinase 1
- Mitogen-activated protein kinase kinase kinase 13 1
- Mitogen-activated protein kinase kinase kinase 10 1
- Mitogen-activated protein kinase kinase kinase 11 1
Publications 1▿
- Blood 114: 2984-92 (2009) 360
Institutions 1▿
- Ambit Biosciences 360
Affinity: 15 to 7.5E+5 nM▿
- IC50 1
- Kd 359
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 1