BDBM50310324 CHEMBL589515::Phe-D-Phe-Arg-Trp-NH2

SMILES N[C@@H](Cc1ccccc1)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O

InChI Key InChIKey=NYOUWNQJCVZGBR-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50310324   

TargetMelanocyte-stimulating hormone receptor(Mouse)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50310324(Phe-D-Phe-Arg-Trp-NH2 | CHEMBL589515)
Affinity DataEC50:  503nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Mouse)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50310324(Phe-D-Phe-Arg-Trp-NH2 | CHEMBL589515)
Affinity DataEC50:  71nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Mouse)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50310324(Phe-D-Phe-Arg-Trp-NH2 | CHEMBL589515)
Affinity DataEC50:  1.19E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Mouse)
The Hebrew University of Jerusalem

Curated by ChEMBL
LigandPNGBDBM50310324(Phe-D-Phe-Arg-Trp-NH2 | CHEMBL589515)
Affinity DataEC50:  143nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed