BDBM50286058 CHEMBL4161506

SMILES [H][C@@]12C[C@]1([H])c1c(C2)c(nn1-c1c[n+]([O-])ccn1)C(=O)NC1(CCC1)C(F)(F)F

InChI Key InChIKey=LSGUAPNQQTXJTL-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50286058   

TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at recombinant human CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant rat CB1 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50286058(CHEMBL4161506)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at recombinant rat CB2 receptor expressed in HEK293 cells assessed as increase in beta arrestin recruitment measured after 2 to 3 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed