BDBM50282652 CHEMBL4159451

SMILES C[C@@H](C(=O)Nc1ncccc1C)c1ccc(c(F)c1)-c1ccccc1

InChI Key InChIKey=NOGZIKCVDIRZRX-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50282652   

TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of FAAH T488A mutant (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 18 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells transfected with empty vector using [3H]AEA as substrate after 18 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 18 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FAAH T488A mutant (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 650nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells transfected with empty vector using [3H]AEA as substrate after 2 hrs by liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50282652(CHEMBL4159451)
Affinity DataIC50: 700nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2020
Entry Details Article
PubMed