BDBM50275924 (S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl)propanoic acid::CHEMBL472451

SMILES OC(=O)[C@H](Cc1ccc(cc1)-c1cccs1)Oc1ccc(Cl)cc1

InChI Key InChIKey=KCXRTOMBQGOLRH-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50275924   

LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  590nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells co-transfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at GAL4-fused PPARgamma (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
LigandPNGBDBM50275924((S)-2-(4-chlorophenoxy)-3-(4-(thiophen-2-yl)phenyl...)
Affinity DataEC50:  589nMAssay Description:Agonist activity at GAL4-fused PPARalpha (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed