BDBM50267948 CHEMBL4097333

SMILES Nc1ccc(cc1)C1=NN(C2CC(Br)=NO2)C(=O)Cc2cc3OCCOc3cc12

InChI Key InChIKey=WXZDBSUEQSNNNB-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50267948   

TargetGlutamate receptor 2(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50267948(CHEMBL4097333)
Affinity DataKi:  3.00E+3nMAssay Description:Antagonist activity at closed state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced curre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2020
Entry Details Article
PubMed
TargetGlutamate receptor 2(Human)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50267948(CHEMBL4097333)
Affinity DataKi:  1.40E+4nMAssay Description:Antagonist activity at open state of GluA2Qflip isoform (unknown origin) expressed in HEK293 cells assessed as reduction in glutamate-induced current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2020
Entry Details Article
PubMed