BDBM50260042 CHEMBL4064534
SMILES CN(C)C\C=C\C(=O)Nc1cc(ccc1C)-n1c2c(ccc3ccc(cc23)-c2cnn(C)c2)ccc1=O
InChI Key InChIKey=JNHXDBIEQOIKLK-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50260042
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full length GST-tagged human PIM2 expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
TargetEpithelial discoidin domain-containing receptor 1(Human)
Dana-Farber Cancer Institute
Curated by ChEMBL
Dana-Farber Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 5.02E+3nMAssay Description:Inhibition of GST-tagged human DDR1 catalytic domain (440 to 876 residues) expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged human DDR2 cytoplasmic domain (427 to 855 residues) expressed in baculovirus expression system by LanthaScreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of recombinant full length His-tagged human PIM1 expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of recombinant full length His-tagged human BMX cytoplasmic domain expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
Affinity DataIC50: 911nMAssay Description:Inhibition of recombinant full length His-tagged human BTK cytoplasmic domain expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair