BDBM50256714 9-phenyl-8-(4-((4-(5-(pyridin-2-yl)-1H-1,2,4-triazol-3-yl)piperidin-1-yl)methyl)phenyl)-[1,2,4]triazolo[3,4-f][1,6]naphthyridin-3-amine::CHEMBL499555
SMILES Nc1nnc2c3cc(-c4ccccc4)c(nc3ccn12)-c1ccc(CN2CCC(CC2)c2nnc([nH]2)-c2ccccn2)cc1
InChI Key InChIKey=UVESBJXBNNCHGR-UHFFFAOYSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50256714
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of SGKMore data for this Ligand-Target Pair
Affinity DataIC50: 47.7nMAssay Description:Inhibition of Akt2 by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18.1nMAssay Description:Inhibition of Akt1 by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.32E+3nMAssay Description:Inhibition of human ERG expressed in HEK cells by competitive radioligand binding assayMore data for this Ligand-Target Pair