BDBM50251902 CHEMBL479405::ethyl 2-(3-hydroxy-2-(2-(phenylsulfonyl)acetamido)-2,3-dihydrothiazol-4-yl)acetate

SMILES CCOC(=O)Cc1csc(=NC(=O)CS(=O)(=O)c2ccccc2)n1O

InChI Key InChIKey=PCWNRXQAFWVYIE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50251902   

TargetEgl nine homolog 1(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50251902(ethyl 2-(3-hydroxy-2-(2-(phenylsulfonyl)acetamido)...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human PHD2 assessed as hydroxylation of Pro564 in human HIF-1alpha by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed