BDBM50247946 2-(1-(4-methyl-3-(trifluoromethyl)phenyl)-1H-1,2,3-triazol-4-yl)-N-(pyridin-4-ylmethyl)aniline::CHEMBL523320

SMILES Cc1ccc(cc1C(F)(F)F)-n1cc(nn1)-c1ccccc1NCc1ccncc1

InChI Key InChIKey=RPXAVKZRWOMBEP-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50247946   

LigandPNGBDBM50247946(2-(1-(4-methyl-3-(trifluoromethyl)phenyl)-1H-1,2,3...)
Affinity DataIC50: 140nMAssay Description:Inhibition of VEGFR2 by HTRF assay in presence of 2 uM ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50247946(2-(1-(4-methyl-3-(trifluoromethyl)phenyl)-1H-1,2,3...)
Affinity DataIC50: 110nMAssay Description:Inhibition of VEGFR1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50247946(2-(1-(4-methyl-3-(trifluoromethyl)phenyl)-1H-1,2,3...)
Affinity DataIC50: 180nMAssay Description:Inhibition of VEGF-induced phosphorylation of VEGFR2 by cell-based ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed