BDBM50244098 2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2,2,2-trifluoroethyl)-1H-benzo[d]imidazole-5-carboxamide::CHEMBL510854

SMILES CCOc1ccc(Cc2nc3cc(ccc3n2CC2CC2)C(=O)N(CC(F)(F)F)CC(F)(F)F)cc1

InChI Key InChIKey=NIKRJWCSBDCYRW-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50244098   

TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at cloned human CB2 receptor in Sf9 cells assessed as stimulation of [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataKi:  4.53E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed