BDBM50242522 CHEMBL4061297

SMILES Nc1nc(NCc2ccc(Cl)cc2)c2c(n1)[nH]c1ccc(O)cc21

InChI Key InChIKey=VRMWGDJTEVKHID-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50242522   

TargetEpidermal growth factor receptor(Human)
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50242522(CHEMBL4061297)
Affinity DataKi:  80nMAssay Description:Inhibition of EGFR (unknown origin) using poly(Glu,Tyr)4:1 as substrate in presence of [gamma-33P]-ATP after 60 mins by scintillation counting analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2019
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50242522(CHEMBL4061297)
Affinity DataKi:  3.24E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using poly(Glu,Tyr)4:1 as substrate in presence of [gamma-33P]-ATP after 60 mins by scintillation counting anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2019
Entry Details Article
PubMed