BDBM50241812 CHEMBL4074425
SMILES [H][C@@]1([#6]-[#6][C@@]2([H])\[#6](-[#6]-[#6]-[#6][C@]12[#6])=[#6]\[#6]=[#6]-1\[#6]-[#6@@H](-[#8])-[#6](=[#6])-[#6@H](-[#8])-[#6]-1)[#6@H](-[#6])-[#6@@H](-[#6]-[#6]-[#6]-[#6])-[#6]-[#6]C([#8])(c1ccc(-[#8])cc1)c1ccc(-[#8])cc1
InChI Key InChIKey=NHRJCHGJKDYMPX-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50241812
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human vitamin D receptor expressed in HEK293 cells assessed as inhibition of 1,25D3-induced transactivation after 16 hrs by du...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-1,25-(OH)2D3 from N-terminal GST-tagged human recombinant vitamin D receptor ligand binding domain expressed in Escherichia coli...More data for this Ligand-Target Pair