BDBM50236550 CHEMBL4105239
SMILES Oc1ccc(cc1)-c1c[nH]c2ncc(cc12)C(=O)Nc1cccc(O)c1
InChI Key InChIKey=DPSFKKBIIZTWDA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50236550
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 847nMAssay Description:Inhibition of DYRK2 (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataEC50: 3.40E+4nMAssay Description:Inhibition of CLK1 (unknown origin) using KKGRSRSRSRSRSR as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of DYRK1B (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair