BDBM50236542 CHEMBL4088888
SMILES CS(=O)(=O)Nc1ccc(cc1)-c1cnc2[nH]cc(-c3ccc(O)cc3)c2c1
InChI Key InChIKey=KOMXYYABYRRJBD-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50236542
TargetDual specificity protein kinase CLK1(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataEC50: 4.40E+4nMAssay Description:Inhibition of CLK1 (unknown origin) using KKGRSRSRSRSRSR as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 724nMAssay Description:Inhibition of DYRK2 (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of DYRK1B (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair