BDBM50234543 CHEMBL4069973

SMILES Cc1ccccc1-c1ccc2n(nc(F)c2c1)-c1cc(F)c(cc1Cl)C(=O)NS(C)(=O)=O

InChI Key InChIKey=RJFMXHKHXJIREK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50234543   

TargetSodium channel protein type 9 subunit alpha(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50234543(CHEMBL4069973)
Affinity DataIC50: 60nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inhibition of peak current after 50 secs by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2019
Entry Details Article
PubMed