BDBM50233352 CHEMBL4100647

SMILES CC1(C)OOC2(CCC(CC2)C(=O)Nc2ccc3ncnc(Nc4cccc(Cl)c4)c3c2)OO1

InChI Key InChIKey=YEOQLUSHLPPCDY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50233352   

TargetEpidermal growth factor receptor(Human)
Soochow University

Curated by ChEMBL
LigandPNGBDBM50233352(CHEMBL4100647)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GST-tagged EGFR cytoplasmic domain (668 to 1210 residues) expressed in baculovirus expression system by Z'-Lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2019
Entry Details Article
PubMed