BDBM50232630 CHEMBL4062339

SMILES CC1(CC1)OC(=O)N1CCC(CC1)[C@H]1C[C@H]1CCOc1ccc(CC(=O)N2CCC2)c(F)c1

InChI Key InChIKey=HLZBPMJWXRSCQF-UHFFFAOYSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50232630   

LigandPNGBDBM50232630(CHEMBL4062339)
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human ERG by PatchXpress methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
LigandPNGBDBM50232630(CHEMBL4062339)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase in intracellular cAMP level after 60 mins by HTRF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
LigandPNGBDBM50232630(CHEMBL4062339)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed
LigandPNGBDBM50232630(CHEMBL4062339)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP level after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2019
Entry Details Article
PubMed