BDBM50232136 CHEMBL428946::N-(5-fluoro-2,3-dihydro-1H-inden-1-yl)-N'-1H-indazol-4-ylurea

SMILES Fc1ccc2C(CCc2c1)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=JBNOOOTYPGAENR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232136   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232136(N-(5-fluoro-2,3-dihydro-1H-inden-1-yl)-N'-1H-indaz...)Copy SMILESCopy InChI

Affinity DataIC50: 52nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
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