BDBM50232133 CHEMBL401128::N-1H-indazol-4-yl-N'-(5-piperidin-1-yl-2,3-dihydro-1H-inden-1-yl)urea

SMILES O=C(NC1CCc2cc(ccc12)N1CCCCC1)Nc1cccc2[nH]ncc12

InChI Key InChIKey=SVYGRCSOIPQXGO-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232133   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232133(N-1H-indazol-4-yl-N'-(5-piperidin-1-yl-2,3-dihydro...)Copy SMILESCopy InChI

Affinity DataIC50: 14nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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