BDBM50232130 1-(4-tert-butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea::CHEMBL251931

SMILES CC(C)(C)c1cccc2C(CCc12)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=JONVCMQRFWSVMA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232130   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232130(1-(4-tert-butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-i...)Copy SMILESCopy InChI

Affinity DataIC50: 14nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL