BDBM50229206 CHEMBL253310::N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-2-(4-(trifluoromethyl)phenyl)thiazole-5-carboxamide

SMILES Cc1nc(sc1C(=O)NCc1ccc(NS(=O)(=O)C(F)(F)F)cc1)-c1ccc(cc1)C(F)(F)F

InChI Key InChIKey=RBFXKVXGGZSKSM-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50229206   

TargetPeroxisome proliferator-activated receptor delta(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at mouse PPARdelta assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse PPARalpha assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50229206(N-(4-(trifluoromethylsulfonamido)benzyl)-4-methyl-...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at mouse PPARgamma assessed as receptor activation by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed