BDBM50223446 CHEMBL389147::c[Tyr-Tyr-Asp-Glu-Gly-Leu-Glu-Glu]-NH2::c[YYDEGLEE]-NH2

SMILES CC(C)C[C@@H]1NC(=O)CNC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)CC[C@H](NC(=O)[C@H](CCC(O)=O)NC1=O)C(N)=O

InChI Key InChIKey=FRCBDVBWQMWQOW-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50223446   

TargetVascular endothelial growth factor receptor 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50223446(c[Tyr-Tyr-Asp-Glu-Gly-Leu-Glu-Glu]-NH2 | c[YYDEGLE...)
Affinity DataIC50: 3.99E+4nMAssay Description:Displacement of biotinylated VEGF165 from human recombinant VEGFR1 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50223446(c[Tyr-Tyr-Asp-Glu-Gly-Leu-Glu-Glu]-NH2 | c[YYDEGLE...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of biotinylated VEGF165 binding to human recombinant VEGFR1 domain 1 to 3 by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50223446(c[Tyr-Tyr-Asp-Glu-Gly-Leu-Glu-Glu]-NH2 | c[YYDEGLE...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of biotinylated VEGF165 binding to human recombinant VEGFR1 extracellular domain by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed