BDBM50211541 (3S,4R)-N-(2-fluorobenzyl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide::CHEMBL228277::rac-trans-N-(2-fluorobenzyl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethylchroman-6-carboxamide

SMILES CCN(Cc1ccccc1F)C(=O)c1ccc2OC(C)(C)[C@@H](O)[C@H](NS(=O)(=O)c3ccc(CC)cc3)c2c1

InChI Key InChIKey=RDQVJCDDJXYHEK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50211541   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50211541(rac-trans-N-(2-fluorobenzyl)-N-ethyl-4-(4-ethylphe...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50211541(rac-trans-N-(2-fluorobenzyl)-N-ethyl-4-(4-ethylphe...)
Affinity DataIC50: 172nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells assessed as blockade of ultra rapidly activating potassium current by voltage clamp t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed