BDBM50200794 CHEMBL216407::N-(2-(piperazin-1-ylmethyl)quinolin-6-yl)-2-(4-(trifluoromethyl)phenoxy)acetamide

SMILES FC(F)(F)c1ccc(OCC(=O)Nc2ccc3nc(CN4CCNCC4)ccc3c2)cc1

InChI Key InChIKey=OPXXNROYPUXCTG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50200794   

TargetMelanin-concentrating hormone receptor 1(Human)
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50200794(N-(2-(piperazin-1-ylmethyl)quinolin-6-yl)-2-(4-(tr...)
Affinity DataIC50: 122nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from MCH-R1 expressing cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed