BDBM50197624 2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-(trifluoromethyl)phenyl)isoxazol-5-yl)methyl)ethanamine::CHEMBL227532

SMILES Cc1ccc(N2CCN(CCNCc3cc(no3)-c3ccccc3C(F)(F)F)CC2)c(C)c1

InChI Key InChIKey=SQEFMAJJBYCCFF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50197624   

TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50197624(2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of alpha-1G T-type calcium channel expressed in HEK293 cells by electrophysiological methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed