BDBM50185944 CHEMBL208472::N-(1-(4-fluorophenyl)-3-(thiophen-2-yl)-1H-pyrazol-5-yl)-3,5-bis(trifluoromethyl)benzenesulfonamide::N-[1-(4-FLUOROPHENYL)-3-(2-THIENYL)-1H-PYRAZOL-5-YL]-3,5-BIS(TRIFLUOROMETHYL)BENZENESULFONAMIDE

SMILES Fc1ccc(cc1)-n1nc(cc1NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)-c1cccs1

InChI Key InChIKey=BQSKQGGQDUBLNS-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50185944   

TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185944(N-(1-(4-fluorophenyl)-3-(thiophen-2-yl)-1H-pyrazol...)
Affinity DataEC50:  0.780nMAssay Description:Effect on Gal4/PPAR-gamma-LBD construct transactivation in Huh7 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50185944(N-(1-(4-fluorophenyl)-3-(thiophen-2-yl)-1H-pyrazol...)
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]rosiglitazone from PPARgamma by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed