BDBM50178616 CHEMBL3814423

SMILES c1n[nH]c2c1c1c3ccccc3[nH]c1c1[nH]c3ccccc3c21

InChI Key InChIKey=QPVVONUJDZMFFK-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50178616   

TargetSerine/threonine-protein kinase pim-1(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50178616(CHEMBL3814423)
Affinity DataIC50: 150nMAssay Description:Inhibition of human full length (His)6-tagged Pim-1 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-2(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50178616(CHEMBL3814423)
Affinity DataIC50: 590nMAssay Description:Inhibition of human full length GST-tagged Pim-2 expressed in Escherichia coli using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]ATP-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
University of Clermont Auvergne

Curated by ChEMBL
LigandPNGBDBM50178616(CHEMBL3814423)
Affinity DataIC50: 22nMAssay Description:Inhibition of human full length (His)6-tagged Pim-3 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details Article
PubMed