BDBM50164405 CHEMBL3800532

SMILES CCN(Cc1cc(=O)n2nc(C)sc2n1)c1ccc(F)cc1

InChI Key InChIKey=GYQFNGUZPFMLGJ-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50164405   

TargetGlutamate receptor 2(Human)
Pharmaron-Beijing

Curated by ChEMBL
LigandPNGBDBM50164405(CHEMBL3800532)
Affinity DataEC50:  3.30E+3nMAssay Description:Positive allosteric modulation of human GluA2 AMPAR flip isomer expressed in Dox-inducible cells measured every 5 mins by BD calcium indicator dye ba...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Pharmaron-Beijing

Curated by ChEMBL
LigandPNGBDBM50164405(CHEMBL3800532)
Affinity DataEC50:  900nMAssay Description:Positive allosteric modulation of GluN1/GluN2A NMDAR (unknown origin) expressed in Dox-inducible cells measured every 5 mins by BD calcium indicator ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor 2(Human)
Pharmaron-Beijing

Curated by ChEMBL
LigandPNGBDBM50164405(CHEMBL3800532)
Affinity DataEC50:  830nMAssay Description:Positive allosteric modulation of human GluA2 AMPAR flop isomer expressed in Dox-inducible cells measured every 5 mins by BD calcium indicator dye ba...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed