BDBM50148462 CHEMBL3770886

SMILES CC(C)c1ccc(cc1)S(=O)(=O)Nc1ccc2n(C)c(=O)n(C)c2c1

InChI Key InChIKey=NTEOEJNZLOGVBX-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50148462   

TargetTranscription intermediary factor 1-alpha(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148462(CHEMBL3770886)
Affinity DataIC50: 3.45E+3nMAssay Description:Inhibition of N-terminal His6-SUMO-1-tagged recombinant human TRIM24 bromodomain expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells by Alpha Scr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2017
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148462(CHEMBL3770886)
Affinity DataIC50: 420nMAssay Description:Inhibition of BRPF1B (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2017
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50148462(CHEMBL3770886)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of BRPF2 BRD1 (unknown origin) by Alpha Screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2017
Entry Details Article
PubMed