BDBM50136491 5-Methoxy-4,9-dihydro-3H-beta-carboline::CHEMBL6591

SMILES COc1cccc2[nH]c3C=NCCc3c12

InChI Key InChIKey=UXOCVYNVGBOVRY-UHFFFAOYSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50136491   

Target5-hydroxytryptamine receptor 2C(Human)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  65nMAssay Description:Binding affinity to 5-HT2C (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  75nMAssay Description:Binding affinity towards cloned rat 5-hydroxytryptamine 2C receptor from fundus tissue by [3H]mesulergine displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  330nMAssay Description:Binding affinity at alpha-2 adrenergic receptors of rat.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  470nMAssay Description:Binding affinity towards cloned rat 5-hydroxytryptamine 2A receptor by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136491(5-Methoxy-4,9-dihydro-3H-beta-carboline | CHEMBL65...)
Affinity DataKi:  500nMAssay Description:Binding affinity for rat 5-hydroxytryptamine 2A receptor using [3H]DOBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed