BDBM50119380 CHEMBL25236::CHEMBL540612::N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-2-naphthamide::Naphthalene-2-carboxylic acid {4-[4-(2-methoxy-phenyl)-piperazin-1-yl]-butyl}-amide
SMILES COc1ccccc1N1CCN(CCCCNC(=O)c2ccc3ccccc3c2)CC1
InChI Key InChIKey=MNHDKMDLOJSCGN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 72 hits for monomerid = 50119380
Affinity DataEC50: 1.80nMAssay Description:Intrinsic activity in mitogenesis assay using Dopamine receptor D3 expressing CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration for Dopamine receptor D3 was determined in monkeysMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human dopamine D3 receptor expressed in human U2OS cells assessed as inhibition of pramipexole-stimulated beta-arrestin recrui...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Mitogenic stimulation in CHO cells expressing human Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Mitogenic stimulation in CHO cells expressing human Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Mitogenic stimulation in NG 108-15 cells expressing human D3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]nemonapride from Rattus norvegicus (rat) chimeric dopamine D2 trunk/D2 tail receptor transfected in african green monkey COS7 cel...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]nemonapride from Rattus norvegicus (rat) wild type dopamine D2 receptor transfected in african green monkey COS7 cells after 1 hr...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Partial agonist intrinsic activity at dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.720nMAssay Description:Displacement of [3H]nemonapride from Rattus norvegicus (rat) chimeric dopamine D3 trunk/D3 tail receptor transfected in african green monkey COS7 cel...More data for this Ligand-Target Pair
Affinity DataEC50: 49nMAssay Description:Effective concentration from [3H]thymidine uptake assay in CHO10001 cells expressing human Dopamine receptor D4.2More data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Displacement of [3H]nemonapride from Rattus norvegicus (rat) wild type dopamine D3 receptor transfected in african green monkey COS7 cells after 1 hr...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Effective concentration in [3H]thymidine uptake assay by CHO dhfr- mutant cells expressing human D3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Intrinsic activity at human D3 receptor expressed in CHO dhfr- cells assessed as rate of [3H]thymidine incorporation by mitogenesis assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]-IABN from human dopamine D3 receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Inhibition of [3H]YM-09151-2 binding to human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Binding affinity for human dopamine receptor D3 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:Binding affinity for rat striatum Dopamine receptor D3 (sf9 cells) by [3H]7-OH-DPAT displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of [3H]-PD 128907 binding to Dopamine receptor D3 in rat ventral striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity D3 [3H]-PD 128907 receptor was determined using caudate-putamen of adult male Spragueo=Dawley ratsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity towards dopamine D3 receptor in ventral striatal membranes of sprague-dawley rat brain by using [3H]-PD 128907 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]R-(+)-7-OHDPAT from dopamine D3 receptor in Sprague-Dawley rat ventral striatum after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D3 expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]spiperone from human D3 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for human Dopamine receptor D3 by [3H]- spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]spiroperidol from human cloned dopamine D3 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.75nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]-N-methylspiperone from recombinant human D3 receptor (unknown origin) measured after 90 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]spiroperidol from cloned human dopamine receptor D3 in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]-prazosin from human ADRA1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: <10nMAssay Description:Partial agonist activity at D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 20.2nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Human)
University of North Carolina At Chapel Hill
Curated by ChEMBL
University of North Carolina At Chapel Hill
Curated by ChEMBL
Affinity DataKi: 33.1nMAssay Description:Displacement of [3H]LSD from human cloned 5HT2B receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 33.6nMAssay Description:Displacement of [125I]-IABN from human dopamine D2L receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity for human Dopamine receptor D4 by [3H]- spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [3H]spiperone binding to human dopamine receptor D4.4 expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]spiperone from human D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity for rat cortex alpha-1 adrenergic receptor by inhibition of [3H]prazosin bindingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Binding affinity for human dopamine receptor D2 by displacing [125I]iodosulpiride expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Inhibition of [3H]YM-09151-2 binding to human Dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity for rat striatum Dopamine receptor D2 by [3H]spiperone displacement.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of [125I]ABN from human dopamine D2L receptor expressed in HEK293 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Human)
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
National Institute On Drug Abuse-Intramural Research Program
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK293 cell membrane measured after 50 mins by competitive radioligand binding an...More data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Displacement of [3H]- 8-OH-DPAT from porcine 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor of porcine cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity towards porcine serotonin receptor 5-HT1A using [3H]8-OH-DPATMore data for this Ligand-Target Pair