BDBM50100750 CHEMBL410824::Des-AA1,2-[DTrp8]-SRIF

SMILES C[C@@H](O)[C@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](N)CSSCC(NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)[C@@H](C)O)C(O)=O

InChI Key InChIKey=HUGAAIZUHOUHDU-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50100750   

TargetSomatostatin receptor type 3(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100750(Des-AA1,2-[DTrp8]-SRIF | CHEMBL410824)
Affinity DataIC50: 4.30nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100750(Des-AA1,2-[DTrp8]-SRIF | CHEMBL410824)
Affinity DataIC50: 5.40nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 2(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100750(Des-AA1,2-[DTrp8]-SRIF | CHEMBL410824)
Affinity DataIC50: 0.330nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 4(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100750(Des-AA1,2-[DTrp8]-SRIF | CHEMBL410824)
Affinity DataIC50: 3.5nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 5(Human)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50100750(Des-AA1,2-[DTrp8]-SRIF | CHEMBL410824)
Affinity DataIC50: 16.7nMAssay Description:Tested for ability to bind to 20 uM thick cryostat sections of a membrane pellet of cells transfected with human cloned somatostatin (sst) receptor s...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed