BDBM50095314 CHEMBL3589893

SMILES CC(=O)Nc1ccc(c(N)n1)-c1cc(Cl)cc(Cl)c1Cl

InChI Key InChIKey=WFMLWHWVTGVADY-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50095314   

LigandPNGBDBM50095314(CHEMBL3589893)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human Nav1.2 expressed in SHSY5Y cells assessed as reduction in blue fluorescent signal by VSP-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
LigandPNGBDBM50095314(CHEMBL3589893)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human Nav1.3 expressed in SHSY5Y cells assessed as reduction in blue fluorescent signal by VSP-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
LigandPNGBDBM50095314(CHEMBL3589893)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human Nav1.7 expressed in SHSY5Y cells assessed as reduction in blue fluorescent signal by VSP-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
LigandPNGBDBM50095314(CHEMBL3589893)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Nav1.8 expressed in HEK293 cells assessed as reduction in blue fluorescent signal by VSP-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed