BDBM50092833 4-(3-Phenoxy-propyl)-1H-imidazole with (0.95M)oxalic acid::CHEMBL112951::CHEMBL128923

SMILES C(COc1ccccc1)Cc1cnc[nH]1

InChI Key InChIKey=DOOCQHQHBHNOGX-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50092833   

TargetHistamine H3 receptor(Rat)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50092833(CHEMBL128923 | CHEMBL112951 | 4-(3-Phenoxy-propyl)...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to rat Histamine H3 receptor in CHO-K1 cells using [125I]iodoproxyfan as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50092833(CHEMBL128923 | CHEMBL112951 | 4-(3-Phenoxy-propyl)...)
Affinity DataKi:  27nMAssay Description:Inhibition of [125I]iodoproxyfan binding to human histamine H3 receptor of CHO-K1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50092833(CHEMBL128923 | CHEMBL112951 | 4-(3-Phenoxy-propyl)...)
Affinity DataKi:  55nMAssay Description:In vitro inhibitory activity against histamine H3 receptor using [3H]histamine as radioligand from rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50092833(CHEMBL128923 | CHEMBL112951 | 4-(3-Phenoxy-propyl)...)
Affinity DataKi:  55nMAssay Description:Effect on histamine H3 receptors in vitro, on synaptosomes of rat cerebral cortex for the release of [3H]histamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2012
Entry Details Article
PubMed