BDBM50083446 1-(3H-Imidazol-4-ylmethyl)-4-(naphthalene-1-sulfonyl)-7-phenyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine::CHEMBL151362

SMILES O=S(=O)(N1CCN(Cc2cnc[nH]2)c2ccc(cc2C1)-c1ccccc1)c1cccc2ccccc12

InChI Key InChIKey=NKVDSSYZHNHJPX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50083446   

TargetDimer of Protein farnesyltransferase subunit beta(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50083446(1-(3H-Imidazol-4-ylmethyl)-4-(naphthalene-1-sulfon...)
Affinity DataIC50: 4.26E+5nMAssay Description:Inhibitory activity against human purified recombinant farnesyltransferase (hFT)More data for this Ligand-Target Pair
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PubMed