BDBM50083445 2-[1-(3H-Imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-benzo[e][1,4]diazepine-4-sulfonyl]-benzoic acid methyl ester::CHEMBL149923

SMILES COC(=O)c1ccccc1S(=O)(=O)N1CCN(Cc2cnc[nH]2)c2ccccc2C1

InChI Key InChIKey=OHMRZXBSMHSGPK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50083445   

TargetDimer of Protein farnesyltransferase subunit beta(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50083445(2-[1-(3H-Imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-b...)
Affinity DataIC50: 720nMAssay Description:Inhibitory activity against human purified recombinant farnesyltransferase (hFT)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed