BDBM50078630 CHEMBL4296718

SMILES Cn1cc(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(cc2)C#N)cn1

InChI Key InChIKey=RRZVGDGTWNQAPW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50078630   

TargetBromodomain adjacent to zinc finger domain protein 2A(Human)
Cancer Research Uk Cancer Therapeutics Unit

Curated by ChEMBL
LigandPNGBDBM50078630(CHEMBL4296718)
Affinity DataIC50: 136nMAssay Description:Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Human)
Cancer Research Uk Cancer Therapeutics Unit

Curated by ChEMBL
LigandPNGBDBM50078630(CHEMBL4296718)
Affinity DataIC50: 174nMAssay Description:Displacement of H3K14Ac from BAZ2B (unknown origin) preincubated for 30 mins with non-biotinylated peptide followed by addition of biotinylated pepti...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed