BDBM50072632 (S)-2-[2-({(S)-2-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetylamino]-3-methyl-pentyl}-benzyl-amino)-acetylamino]-4-methylsulfanyl-butyric acid::CHEMBL112917
SMILES CCC(C)[C@@H](CN(CC(=O)N[C@@H](CCSC)C(O)=O)Cc1ccccc1)NC(=O)CSc1nc2ccccc2[nH]1
InChI Key InChIKey=MHPGTFOKNTYHDW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50072632
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair