BDBM50057796 CHEMBL3326188

SMILES CCCCCc1ccc(cc1)-c1ccoc1C(=O)NNC(=O)c1ccc(O)c(c1)[N+]([O-])=O

InChI Key InChIKey=XOVVMEVNXYGYEG-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50057796   

TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 9.60E+3nMAssay Description:Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 292nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in human hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of GLP-1R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed