BDBM50055013 6-(3-Chloro-phenyl)-2,3,4,6-tetrahydro-pyrimido[2,1-a]isoindol-6-ol::9-(3-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-fluoren-9-ol::CHEMBL133786

SMILES OC1(N2CCCN=C2c2ccccc12)c1cccc(Cl)c1

InChI Key InChIKey=ZTSMFSRRQVVDJN-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50055013   

TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055013(9-(3-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]WIN-35428 binding to the dopamine transporter in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055013(9-(3-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of [3H]dopamine uptake at the dopamine transporter in rat striatal tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Drew University

Curated by ChEMBL
LigandPNGBDBM50055013(9-(3-Chloro-phenyl)-1,2,3,9-tetrahydro-4,9a-diaza-...)
Affinity DataIC50: 1nMAssay Description:Ability to displace [3H]WIN-35428 from dopamine transporter in rat caudate putamen tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed